Overview

Definition:
-Asthma biologic selection in pediatrics involves using targeted therapies, primarily monoclonal antibodies, to treat severe or uncontrolled asthma that is refractory to conventional inhaled corticosteroids and long-acting beta-agonists
-This approach is guided by specific phenotypic characteristics of the child's asthma, such as eosinophilic inflammation or allergic sensitization.
Epidemiology:
-Asthma is the most common chronic respiratory disease in children, affecting approximately 6-9% globally
-Severe asthma accounts for 5-10% of childhood asthma cases
-Phenotyping allows for more precise management of these complex cases, which are associated with higher healthcare utilization and poorer quality of life.
Clinical Significance:
-Identifying distinct asthma phenotypes is crucial for optimizing treatment strategies
-Phenotype-based selection of biologics offers a paradigm shift from a one-size-fits-all approach, leading to improved symptom control, reduced exacerbations, decreased oral corticosteroid dependence, and enhanced overall well-being in children with severe asthma
-This is critical for residents preparing for DNB and NEET SS examinations.

Phenotypes And Biologic Targets

Allergic Asthma Type 2 High:
-Characterized by elevated IgE, eosinophils, and atopy
-Targeted by anti-IgE (omalizumab) and anti-IL-5/5R (mepolizumab, reslizumab, benralizumab).
Eosinophilic Asthma Type 2 High:
-Defined by persistent sputum eosinophilia (>=300 cells/µL) or blood eosinophilia (>=400 cells/µL) independent of atopy
-Targeted by anti-IL-5/5R agents.
Other Phenotypes: Includes neutrophilic asthma and paucigranulocytic asthma, for which current biologic options are less established, though research is ongoing for other targets like TSLP.

Biologic Agents In Pediatrics

Omalizumab Anti Ige:
-Indicated for moderate-to-severe persistent allergic asthma in children aged 6 years and older with sensitization to perennial allergens
-Administered subcutaneously every 2-4 weeks
-Dosage based on IgE levels and body weight.
Anti Il 5 Inhibitors:
-Mepolizumab: Approved for severe eosinophilic asthma in children aged 12 years and older
-Reslizumab: Approved for severe eosinophilic asthma in adults (less data in pediatrics)
-Benralizumab: Approved for severe eosinophilic asthma in children aged 12 years and older
-All administered subcutaneously every 4-8 weeks.
Anti Il 4 Receptor Alpha Inhibitors:
-Dupilumab: Approved for moderate-to-severe atopic asthma in children aged 6 years and older with type 2 inflammation
-Blocks both IL-4 and IL-13 signaling
-Administered subcutaneously every 2-4 weeks.

Patient Selection And Assessment

Diagnostic Evaluation:
-Confirm diagnosis of severe asthma
-Assess for persistent symptoms despite optimal conventional therapy
-Evaluate for type 2 inflammation markers: elevated IgE, blood/sputum eosinophilia, atopy (skin prick tests or specific IgE).
Exclusion Criteria:
-Rule out alternative diagnoses or contributing factors such as poorly controlled rhinosinusitis, GERD, obesity, vocal cord dysfunction, or environmental exposures
-Ensure adherence to prescribed inhaled therapies.
Monitoring Response:
-Assess treatment response after 3-6 months using validated asthma control questionnaires (e.g., ACT/cACT), spirometry (FEV1), exacerbation rates, and oral corticosteroid reduction
-Discontinue if no significant benefit is observed.

Management Considerations And Follow Up

Initiation And Dosing:
-Biologics are typically initiated by a pediatric pulmonologist
-Dosing is weight-based and/or IgE level-based for omalizumab, and fixed for IL-5 and IL-4/13 inhibitors
-Ensure proper patient and caregiver education on administration and potential side effects.
Adverse Events:
-Common side effects include injection site reactions
-Anaphylaxis is rare but serious, particularly with omalizumab
-Monitor for any new or worsening symptoms, including infections.
Long Term Management:
-Continue with optimal conventional therapy alongside biologics
-Regular follow-up with the pulmonologist is essential to monitor efficacy, safety, and potential need for dose adjustment or discontinuation
-Consider transitioning to adult care when appropriate.

Key Points

Exam Focus:
-Phenotype-based selection is key for severe pediatric asthma
-Type 2 inflammation markers (IgE, eosinophils, atopy) guide choice of omalizumab, anti-IL-5, or anti-IL-4/13 agents
-Know indications, age limits, and common administration routes for each biologic.
Clinical Pearls:
-Always re-evaluate the patient and optimize conventional therapy before initiating biologics
-Consider the burden of disease and patient preferences when discussing treatment options
-Early identification of non-responders is crucial.
Common Mistakes:
-Starting biologics without a clear phenotype or adequate trial of conventional therapy
-Failing to monitor response adequately
-Not excluding alternative diagnoses or exacerbating factors.