Overview

Definition:
-Glucose-6-phosphate dehydrogenase (G6PD) deficiency is an X-linked recessive genetic disorder characterized by a deficiency in the enzyme G6PD
-This enzyme is crucial for the pentose phosphate pathway in red blood cells, which protects them from oxidative stress by producing NADPH
-Without sufficient G6PD, red blood cells are susceptible to hemolysis when exposed to oxidative triggers.
Epidemiology:
-G6PD deficiency is the most common human enzyme defect, affecting an estimated 400 million people worldwide
-It is particularly prevalent in populations from malaria-endemic regions, including parts of Africa, Asia, the Mediterranean, and the Middle East
-In India, its prevalence varies significantly by region, with higher rates observed in certain communities
-Neonatal jaundice is a common manifestation in newborns with G6PD deficiency, especially in genetically predisposed populations.
Clinical Significance:
-G6PD deficiency is clinically significant due to the risk of acute hemolytic anemia triggered by certain drugs, foods, and infections
-In neonates, it is a leading cause of severe, unconjugated hyperbilirubinemia and kernicterus
-Understanding its triggers and management is vital for preventing life-threatening complications and is a frequent topic in DNB and NEET SS pediatrics examinations.

Neonatal Jaundice

Introduction:
-Neonatal jaundice is a common condition, but severe hyperbilirubinemia in G6PD deficient neonates poses a significant risk
-This deficiency impairs the red blood cell's ability to handle oxidative stress, leading to premature destruction (hemolysis).
Pathophysiology:
-In neonates, the liver's bilirubin conjugation capacity is immature
-In G6PD deficient infants, oxidative stress from various sources can trigger rapid hemolysis, overwhelming the already limited conjugation pathway
-This leads to a rapid rise in unconjugated bilirubin, potentially exceeding safe levels.
Triggers In Neonates:
-Triggers in neonates are often less clear-cut than in older individuals but can include: Maternal medications passed through breast milk
-Certain topical agents applied to the neonate
-Neonatal infections
-Hypothermia or acidosis
-Oxytetracycline and nitrofurantoin administered to the neonate.
Clinical Features In Newborns:
-Jaundice typically appears within the first 24-72 hours of life
-The icterus may be severe and progress rapidly
-Signs of hemolysis may include pallor, lethargy, and sometimes mild hepatosplenomegaly
-Severe hyperbilirubinemia can lead to kernicterus, characterized by lethargy, poor feeding, hypotonia, opisthotonos, seizures, and sensorineural hearing loss.

Triggers Of Hemolysis

Drug Induced Hemolysis:
-Certain medications are potent triggers
-Common culprits include: Antimalarials: Primaquine, quinine, chloroquine
-Sulfonamides: Sulfamethoxazole, sulfasalazine
-Analgesics/Antipyretics: Aspirin (high doses), phenacetin
-Antibiotics: Dapsone, isoniazid, nitrofurantoin, nalidixic acid
-Others: Fava beans (divicine and isouramil), menthol, methylene blue.
Food Induced Hemolysis:
-The most notorious food trigger is the fava bean (Vicia faba), leading to the condition known as "favism." Other legumes may also pose a risk for highly sensitive individuals
-Consumption of uncooked or partially cooked fava beans is particularly dangerous.
Infection Induced Hemolysis:
-Infections, particularly viral hepatitis, infectious mononucleosis, and urinary tract infections, can induce hemolytic crises in G6PD deficient individuals
-The oxidative stress generated by the host's immune response to infection can precipitate hemolysis.
Other Triggers:
-Other less common triggers include diabetic ketoacidosis, severe burns, and exposure to certain chemicals or dyes
-Stressful events and major surgery can also increase oxidative load.

Diagnostic Approach

History Taking:
-A detailed history is crucial, focusing on: Onset and progression of jaundice (in neonates)
-History of similar episodes in the family
-Exposure to potential triggers: medications, fava beans, infections
-Ethnic background
-Maternal medication history during pregnancy and breastfeeding.
Physical Examination:
-In neonates: Assess degree of jaundice (icteric sclera, skin color)
-Check for pallor, lethargy, poor feeding
-Examine for hepatosplenomegaly
-In older children/adults: Look for pallor, jaundice, splenomegaly
-Signs of acute hemolysis: dark urine (hemoglobinuria).
Investigations:
-Screening: Quantitative G6PD assay (most reliable)
-Measure NADPH production by red blood cells
-It is important to note that G6PD levels can be falsely normal during an acute hemolytic episode due to the preferential destruction of older red blood cells with lower G6PD activity
-therefore, testing should ideally be performed 2-3 months after the crisis
-Fluorescent spot test (less sensitive)
-Confirm diagnosis by genetic testing if needed
-For neonatal jaundice: Total and direct bilirubin levels
-Blood group and Coombs test (to rule out other causes of hemolysis)
-Complete blood count with reticulocyte count
-Peripheral smear for bite cells and blister cells (suggestive of G6PD deficiency)
-Liver function tests
-Urinary analysis for hemoglobinuria.
Differential Diagnosis:
-Neonatal jaundice: Physiologic jaundice, breast milk jaundice, ABO/Rh incompatibility, cephalohematoma, sepsis, hypothyroidism, galactosemia, hereditary spherocytosis, other enzyme deficiencies (e.g., pyruvate kinase deficiency)
-Hemolytic anemia in older individuals: Autoimmune hemolytic anemia, hereditary spherocytosis, thalassemia, sickle cell disease, paroxysmal nocturnal hemoglobinuria, drug-induced immune hemolytic anemia.

Management

Neonatal Management:
-Immediate discontinuation of any suspected trigger
-Phototherapy for mild to moderate hyperbilirubinemia
-Exchange transfusion for severe hyperbilirubinemia or signs of kernicterus
-Avoidance of triggering medications and agents
-Close monitoring of bilirubin levels and signs of hemolysis
-Genetic counseling for the family.
Management Of Hemolytic Crisis:
-The cornerstone of management is immediate cessation of the offending trigger (drug, food, etc.)
-Supportive care includes hydration and monitoring vital signs
-Blood transfusions may be required for severe anemia
-Folic acid supplementation can be considered to support red blood cell production, though its role in acute crisis is debated.
Prevention Strategies:
-Patient and family education regarding triggers is paramount
-Provide patients with a list of contraindicated drugs and foods
-Advise caution with herbal remedies and over-the-counter medications
-Encourage prompt medical attention for any signs of infection
-Genetic screening before prescribing certain medications (e.g., primaquine) is recommended in at-risk populations.
Specific Management Considerations:
-Avoidance of methylene blue, which is often used to treat methemoglobinemia but is a potent G6PD trigger
-Use of alternative therapies for malaria in affected individuals
-Careful consideration of drug choices in patients with known G6PD deficiency.

Complications

Early Complications:
-Acute hemolytic anemia
-Severe hyperbilirubinemia leading to kernicterus in neonates
-Acute kidney injury due to hemoglobinuria
-Splenic rupture (rarely).
Late Complications:
-Chronic hemolytic anemia (mild, in some individuals)
-Sensorineural hearing loss (sequela of kernicterus)
-Cholelithiasis (gallstones) due to chronic hemolysis
-Anemia of chronic disease.
Prevention Strategies:
-Primary prevention involves rigorous avoidance of known triggers by affected individuals and their families
-Secondary prevention focuses on prompt recognition and management of hemolytic episodes to prevent severe complications like kernicterus and kidney injury
-Genetic counseling and carrier screening can help.

Prognosis

Factors Affecting Prognosis:
-The severity of the G6PD deficiency genotype
-The type and extent of trigger exposure
-Promptness of diagnosis and management
-Presence of co-existing medical conditions.
Outcomes:
-With proper avoidance of triggers, most individuals with G6PD deficiency live normal lives
-Neonates with G6PD deficiency, if managed promptly, have a good prognosis
-However, delayed diagnosis and treatment of severe hyperbilirubinemia can lead to irreversible neurological damage (kernicterus).
Follow Up:
-Regular follow-up is recommended, especially for neonates who experienced severe hyperbilirubinemia, to monitor for developmental milestones and hearing
-Patients should be educated to inform all healthcare providers about their condition and to carry an identification card detailing their G6PD deficiency and triggers.

Key Points

Exam Focus:
-G6PD deficiency is an X-linked disorder
-Triggers include certain drugs (antimalarials, sulfonamides, dapsone), fava beans, and infections
-Neonatal jaundice can be severe and lead to kernicterus
-G6PD levels can be falsely normal during hemolysis
-Avoidance of triggers is key.
Clinical Pearls:
-Always consider G6PD deficiency in neonates with unexplained severe hyperbilirubinemia, especially from endemic regions
-Educate patients and families thoroughly on trigger avoidance
-Remember to test G6PD levels a few months after an acute hemolytic episode for accurate diagnosis.
Common Mistakes:
-Prescribing known triggering drugs without checking G6PD status
-Misinterpreting normal G6PD levels during an acute hemolytic crisis
-Failing to promptly initiate phototherapy or exchange transfusion for severe neonatal jaundice
-Inadequate patient education regarding trigger avoidance.